Production scientifique de l'équipe Chimie moléculaire

2024

Fluorine 18 complex useful for positron emission tomography, EP24315112.3. F. Dioury, C. San, M. Port, L. Sarda Mantel

M. Lancel, M. Lindgren, C. Monnereau, Z. Amara, "Kinetic Effects in Singlet Oxygen Mediated Oxidations by Immobilized Photosensitizers on Silica" Photochem. Photobiol. Sci. 2024, 23, 79–92

A. Hadj Mohamed, A. Pinon, N. Lagarde, C. Ricco, E. Goya-Jorge, H. Mouhsine, M. Msaddek, B. Liagre, M Sylla-Iyarreta Veitía, "Colorectal Anticancer Activity of a Novel Class of Triazolic Triarylmethane Derivatives", RSC Med. Chem., 2024, Advance Article

2023

M. Lancel, B. Tambosco, Z. Amara, “Photochemical Routes to Artemisinin”, Specialist Periodic Report Photochemistry: Volume 51, Eds. S. Crespi; S. Protti, Royal Society of Chemistry, 2023.

M. Lancel, T. Golisano, C. Monnereau, C. Gomez, M. Port, Z. Amara, “Sustainable Photooxidations using a Sub-ppm Metal-Free Red Light Photocatalyst” ACS Sustainable Chem. Eng. 2023, 11, 15674–15684

M. Lancel, C. Gomez, M. Port, Z. Amara, “Développement de procédés photocatalytiques plus durables : stratégies d’hétérogénéisation de photocatalyseurs homogènes et intensification des procédés en flux continu” Actualité Chimique, 2023, 488, 7-16

Carine San, Benoît Hosten, Nicolas Vignal, Meriem Beddek, Maurice Pillet, Laure Sarda-Mantel, Marc Port, Fabienne Dioury, Optimization of a NODA Derivative Radiofluorination by Al18F Complexation using a Design of Experiments Approach, Chem. Eur. J. 2023, 29, e2023027

Phthalocyanines supported on silica and their use as a photocatalyst. EP23305918.7. Z. Amara, M. Lancel, M. Port, C. Gomez.

M. Lancel, P. Zimberlin, C. Gomez, M. Port, L. Khrouz, C. Monnereau, Z. Amara, Self-Sensitized Photooxidation of Naphthols to Naphthoquinones and the use of Naphthoquinones as Visible Light Photocatalysts in Batch and Continuous Flow Reactors, J. Org. Chem. 2023, 88, 10, 6498–6508 (Special issue "Progress in Photocatalysis for Organic Chemistry")

C. Linger, M. Lancel, M. Port, Evaluation of relative efficiency of PDT photosensitizers in producing hydroxyl radicals and singlet oxygen in aqueous media using a UV–visible spectroscopy pNDA dosage, J. Photochem. Photobiol. B, 2023, 241, 112664

Z. Amara, Pyrroloquinolines, a New Platform for Developing Organic Photosensitizers: When Synthetic Methodology Meets Photophysics, Photochem. Photobiol. 2023, 99, 863-865 (Highlight article).

A. H. Mohamed, A. Pinon, N. Lagarde, E. Goya Jorge, H. Mouhsine, M. Msaddek, B. Liagre, M. Sylla-Iyarreta Veitia. Novel Set of Diarylmethanes to Target Colorectal Cancer : Synthesis, In Vitro and In Silico Studies. Biomolecules, 2023, 13, 54.

J. C. S. Terra, A, Desgranges, Z. Amara, A. Moores, Photocatalysis on magnetic supports for singlet oxygen generation: Role of immobilization and photobleaching, Catalysis Today, 2023, 407, 52-58

2022

Compounds and methods for treating a cytokine mediated disease. WO2022101453 (A1) H. Mouhsine, A. Mascret, M. Port, J-F. Zagury, M. Montès, M. Sylla-Iyarreta Veitía, C. Ricco, D. Cabrera, M. Benchekroun.

B. Rostom, R. Karaky, I. Kassab, M. Sylla-Iyarreta Veitía. Coumarins derivatives and inflammation: Review of their effects on the inflammatory signaling pathways. Eur. J. Pharma, 2022, 922, 174867

F. Dioury, M. Callewaert, C. Cadiou, C. Henoumont, M. Zolinari, S. Laurent, C. Portefaix, M. Port, F. Chuburu, Pyclen-based Gd complex with ionisable side-chain as a contrastophore for the design of hypersensitive MRI nanoprobes: Synthesis and relaxation studies, Results in Chemistry, 2022, 3, 100237

2021

G. Attia, A. Mascret, C. Zerrouki, N. Fourati, M. Sylla-Iyarreta Veitía, M. Port, Data of the quantification of the influence of DMSO concentration on the kinetic of interaction between TNFα and SPD304, Data in Brief, 2021, 39, 107610

M. Lancel, C. Gomez, M. Port, Z. Amara, Performances of Homogeneous and Heterogenized Methylene Blue on Silica under Red Light in Batch and Continuous Flow Photochemical Reactors, Front. Chem. Eng., 2021, 3, 752364

C. Henoumont, G. Hallot, E. Lipani, C. Gomez, R. N. Muller, L. Vander Elst, M. Port, S. Laurent, Characterization of Organic Molecules Grafted to Silica or Bismuth Nanoparticles by NMR, Appl. Nano 2021, 2(4), 330-343

C. Gomez, G. Hallot, S. Laurent, M. Port, Medical Applications of Metallic Bismuth Nanoparticles, Pharmaceutics 2021, 13, 1793

G. Hallot, V. Cagan, S. Laurent, C. Gomez, M. Port, A Greener Chemistry Process Using Microwaves in Continuous Flow to Synthesize Metallic Bismuth Nanoparticles, ACS Sustainable Chem. Eng. 2021, 9, 9177-9187

A. Mascret, H. Mouhsine, G. Attia, D. Cabrera, M. Benchekroun, P. Gizzie, C. Zerrouki, N. Fourati, J-F. Zagury, M. Sylla-Iyarreta Veitía, M. Port, New contributions to the drug profile of TNFα inhibitor SPD304: Affinity, selectivity and ADMET considerations, Eur. J. Pharmacol. 2021, 907, 174285

A. Gellé, G. D. Price, F. Voisard, N. Brodusch, R. Gauvin, Z. Amara, A. Moores, Enhancing Singlet Oxygen Photocatalysis with Plasmonic Nanoparticles, ACS App. Mat. Interfaces, 2021, 13, 35606-35616

A. Zanetti, G. Schwertz, M. Nascimento de Oliveira, M. A. Gomez Fernandez, Z. Amara, J. Cossy, Palladium-Catalyzed Regioselective Allylic Oxidation of Amorphadiene, a Precursor of Artemisinin, J. Org. Chem. 2021, 86, 7603-7608

M. A. Gomez Fernandez, M. Nascimento de Oliveira, A. Zanetti, G. Schwertz, J. Cossy, Z. Amara, Photochemical Hydrothiolation of Amorphadiene and Formal Synthesis of Artemisinin via a Pummerer Rearrangement, Org.Lett. 2021, 23, 5593-5598 (selected as front cover picture)

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E. Goya-Jorge, M. E. Jorge Rodríguez, M. Sylla-Iyarreta Veitía, R. M. Giner, Plant Occurring Flavonoids as Modulators of the Aryl Hydrocarbon Receptor, Molecules, 2021, 26 (8), 2315

C. Linger, G. Dumy, M. Port, Thérapie Sonodynamique, Techniques de l'ingénieur, 2021, MED2000 v1

M. Devreux, C. Henoumont, F. Dioury, S. Boutry, O. Vacher, L. Vander Elst, M. Port, R. N. Muller, O. Sandre, S. Laurent, Mn2+ Complexes with Pyclen-Based Derivatives as Contrast Agents for Magnetic Resonance Imaging: Synthesis and Relaxometry Characterization, Inorg. Chem. 2021, 60, 3604–3619

2020

Bismuth metallic (0) nanoparticles, process of manufacturinf and uses thereof. WO2020007822 (A1) Port, Marc. Gomez, Catherine. Gauthier Hallot

E. Goya Jorge, C. Rampal, N. Loones, S. J. Barigye, R. Gozalbes, C. Ferroud, M. Sylla-Iyarreta Veitía, R. M. Giner. Targeting the aryl hydrocarbon receptor with a novel set of triarylmethanes. European Journal of Medicinal Chemistry, 2020, 207, 112777.

D. Franchi, Z. Amara, Applications of Sensitized-Semiconductors as Heterogeneous Visible-Light Photocatalysts in Organic Synthesis, ACS Sustain. Chem. Eng. 2020, 8, 15405-15429, Open Access

G. Schwertz, A. Zanetti, M. Nascimento de Oliveira, M. A. Gomez Fernandez, Z. Amara, J. Cossy, Chemo- and Diastereoselective Hydrosilylation of Amorphadiene toward the Synthesis of Artemisinin, J. Org. Chem. 2020, 85, 9607-9613, Open Access

E. Goya-Jorge, F. Abdmouleh, L. E. Carpio, R. M. Giner, M. Sylla-Iyarreta Veitía, Discovery of 2-aryl and 2-pyridinylbenzothiazoles endowed with antimicrobial and aryl hydrocarbon receptor agonistic activities, Eur. J. Pharm. Sci., 2020, 151, 105386

E. Goya-Jorge, R. M. Giner, M. Sylla-Iyarreta Veitía, R. Gozalbes, S. J. Barigye, Predictive modeling of aryl hydrocarbon receptor (AhR) agonism, Chemosphere, 2020, 256, 127068.

J. C. S. Terra, A. Desgranges, C. Monnereau, E. H. Sanchez, J. A. De Toro, Z. Amara, A. Moores, Photocatalysis Meets Magnetism: Designing Magnetically Recoverable Supports for Visible-Light Photocatalysis, ACS Appl. Mater. Interfaces, 2020,12, 24895–24904

M. Russo, Z. Amara, J. Fenneteau, P. Chaumont-Olive, I. Maimouni, P. Tabeling, J. Cossy, Stable Liquid Foams from a New Polyfluorinated Surfactant, Chem. Commun., 2020, 56, 5807-5810

D. Fanfone, D. Stanicki, D. Nonclercq, M. Port, L. Vander Elst, S. Laurent, R. N. Muller, S. Saussez, C. Burtea, Molecular Imaging of Galectin-1 Expression as a Biomarker of Papillary Thyroid Cancer by Using Peptide-Functionalized Imaging Probes, Biology, 2020, 9, 53, Open Access, Special Issue: Molecular Targets and Targeting in Biomedical Sciences

C. Ricco, F. Abdmoulehab, C. Riccobono, L. Guenineche, F. Martin, E. Goya-Jorge, N. Lagarde, B. Liagre, M. BenAli, C. Ferroud, M. ElArbi, M. Sylla-Iyarreta Veitía, Pegylated Triarylmethanes: Synthesis, Antimicrobial Activity, Anti-proliferative Behavior and in Silico Studies, Bioorg. Chem. 2020, 96, 103591

A. Zanetti, P. Chaumont-Olive, G. Schwertz, M. Nascimento de Oliveira, M. A. Gomez Fernandez, Z. Amara, J. Cossy, Crystallization-Induced Diastereoisomer Transformation of Dihydroartemisinic Aldehyde with the Betti Base, Org. Process Res. Dev., 2020, 24, 850–855, Open Access, Special Issue: "A Taste of Current French Organic Chemistry".

V. Blanchard, Z. Asbai, K. Cottet, G. Boissonnat, M. Port, Z. Amara, Continuous Flow Photo-oxidations Using Supported Photocatalysts on Silica, Org. Process Res. Dev., 2020, 24, 822–826, Special Issue: "A Taste of Current French Organic Chemistry".

2019

M. Sylla-Iyarreta Veitía, C. Rampal, C. Ferroud. An Efficient Access to Unsymmetrical Triarylmethanes by Regioselective Friedel-Crafts Hydroxyalkylation. Trends in Organic chemistry, 2019, 20, 1-13

M. Devreux, C. Henoumont, F. Dioury, D. Stanicki, S. Boutry, L. Larbanoix, C. Ferroud, R. N. Muller, S. Laurent, Bimodal Probe for Magnetic Resonance Imaging and Photoacoustic Imaging Based on a PCTA‐Derived Gadolinium(III) Complex and ZW800–1, Eur. J. Inorg. Chem. 2019, 3354–3365

J. Yong-Sang, F. Dioury, V. Meneyrol, I. Ait-Arsa, J-P. Idoumbin, F. Guibbal, J. Patché, F. Gimié, I. Khantalin, J. Couprie, P. Giraud, S. Benard, C. Ferroud, E. Jestin, O. Meilhac, Development, Synthesis, and 68Ga-Labeling of a Lipophilic Complexing Agent for Atherosclerosis PET Imaging, Eur. J. Med. Chem., 2019, 176, 129-134

C. Robic, M. Port, O. Rousseaux, S. Louguet, N. Fretellier, S. Catoen, C. Factor, S. Le Greneur, C. Medina, P. Bourrinet, I. Raynal, J-M. Idée, C. Corot, Physicochemical and Pharmacokinetic Profiles of Gadopiclenol A New Macrocyclic Gadolinium Chelate With High T1 Relaxivity, Invest. Radiol., 2019, 54, 475-484

C. Gomez, G. Hallot, A. Pastor, S. Laurent, E. Brun, C. Sicard-Roselli, M. Port, Metallic Bismuth Nanoparticles: Towards a Robust, Productive and Ultrasound Assisted Synthesis from Batch to Flow-Continuous Chemistry, Ultrason. Sonochem., 2019, 56, 167-173

G. Schwertz, A. Zanetti, M. Nascimento de Oliveira, M. A. Gomez Fernandez, F. Dioury, J. Cossy, Z. Amara, Synthesis of Amorpha-4,11-Diene from Dihydroartemisinic Acid. Tetrahedron, 2019, 75, 743-748

2018

J. Vitku, L. Kolatorova, C. Ricco , C. Ferroud , O. Hennebert, T. Skodova , J. Heracek, L. Starka, The Quantitation of 7β-Hydroxy-Epiandrosterone in the Plasma and Seminal Plasma of Men With Different Degrees of Fertility, Physiol. Res. 2018, 67 (Suppl. 3): S511-S519,

L. Halby, N. Marechal, D. Pechalrieu, V. Cura, D-M. Franchini, C. Faux, F. Alby, N. Troffer-Charlier, S. Kudithipudi, A. Jeltsch, W. Aouadi, E. Decroly, J-C. Guillemot, P. Page, C. Ferroud, L. Bonnefond, D. Guianvarc’h, J. Cavarelli, P. B. Arimondo, Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors. Phil. Trans. R. Soc. B, 2018, 373, 20170072

C. Gomez, G. Hallot, M. Port, Chapter 10, Bismuth metallic nanoparticles, in Inorganic Frameworks as Smart Nanomedicines, edited by Alexandru Mihai Grumezescu,, William Andrew Publishing, 2018, Pages 449-487, ISBN 9780128136614

B. Tambosco, K. Segura, C. Seyrig, D. Cabrera, M. Port, C. Ferroud, Z. Amara, Outer-sphere effects in visible-light photochemical oxidations with immobilized and recyclable ruthenium bipyridyl salts. ACS Catalysis, 2018, 8, 4383-4389

S. Drouet, B. Haider Abbas, A. Falguières, W. Ahmad, S. Khan, C. Ferroud, J. Doussot, J. R. Vanier, E. Lainé, C. Hano, Single Laboratory Validation of a Quantitative Core Shell-Based LC Separation for the Evaluation of Silymarin Variability and Associated Antioxidant Activity of Pakistani Ecotypes of Milk Thistle (Silybum Marianum L.). Molecules, 2018, 23, 904

A. Rayar, N. Lagarde, F. Martin, F. Blanchard, B. Liagre, C. Ferroud, J-F Zagury, M. Montes, M. Sylla-Iyarreta Veitía, New selective cyclooxygenase-2 inhibitors from cyclocoumarol: synthesis, characterization, biological evaluation and molecular modeling. Eur. J. Med. Chem., 2018, 146, 577-587

2017

D. Siverio-Mota, I. Andujar, Y. Marrero-Ponce, R. M. Giner, C. Díaz Mendoza, G. Manjarrez Paba, L. Vicet-Muro, M. L. Cordero-Maldonado, P. A. M de Witte, A. D. Crawford, M. Sylla-Iyarreta Veitía, F. Pérez-Jiménez, V. J. Aran. Anti-Inflammatory activity and cheminformatics analysis of new potent 2-substituted 1-methyl-5-nitroindazolinones. Curr. Top. Med. Chem., 2017, 17, 3236 - 3248

L. Halby, Y. Menon, E. Rilova, D. Pechalrieu, V. Masson, C. Faux, M.A. Bouhlel, M-H. David-Cordonnier, N. Novosad, Y. Aussagues, A. Samson, L. Lacroix, F. Ausseil, L. Fleury, D. Guianvarc'h, C. Ferroud, P. Arimondo, Rational design of bisubstrate-type analogs as inhibitors of DNA methyltransferases in cancer cells, J. Med. Chem., 2017, 60, 4665-4679

J. Jin, S. Guidi, Z. Abada, Z. Amara, M. Selva, M. W. George, M. Poliakoff, Continuous niobium phosphate catalysed Skraup reaction for quinoline synthesis from solketal, Green Chem. 2017, 19, 2439-2447

D. S. Lee, Z. Amara, C. A. Clark, Z. Xu, B. Kakimpa, H. P. Morvan, S. J. Pickering, M. Poliakoff, M. W. George, Continuous photo-oxidation in a vortex reactor: efficient operations using air drawn from the laboratory, Org. Process Res. Dev. 2017, 21, 1042-1050

M. Sylla-Iyarreta Veitía, D. Siverio Mota, V. Lerari, M. Marín, R. M. Giner, L. Vicet Muro, Y. Rivero Guerra, F. Dumas, C. Ferroud, P. A. M. de Witte, A. D. Crawford, V. J. Arán, Y. Marrero Ponce, Fishing Anti-Inflammatories from Known Drugs: In Silico Repurposing, Design, Synthesis and Biological Evaluation of Bisacodyl Analogues, Curr. Top. Med. Chem., 2017, 17, 2866 – 2887,

Rayar A.-M., Lagarde N., Ferroud C., Zagury J.-F., Montes M., Sylla-Iyarreta Veitía M., Update on COX-2 Selective Inhibitors: Chemical Classification, Side Effects and their Use in Cancers and Neuronal Diseases, Curr. Top. Med. Chem., 2017, 17, 1-22.

M. Sylla-Iyarreta Veitía, F. Dumas, A. Duardo-Sánchez, S. Arrasate, Editorial: New Experimental and Computational Tools for Drug Discovery: From Chemistry to Biology. Part-III, Curr. Top. Med. Chem, 2017, 17(30): 3234 – 3235.

M. Sylla-Iyarreta Veitía, F. Dumas, H. González-Díaz. Editorial: New Experimental and Computational Tools for Drug Discovery: From Chemistry to Biology. Part-II, Curr. Top. Med. Chem., 2017, 17(26): 2901 – 2902.

M. Sylla-Iyarreta Veitía, F. Dumas, H. González-Díaz, Editorial: New Experimental and Computational Tools for Drug Discovery: From Chemistry to Biology. Part-I, Curr. Top. Med. Chem., 2017, 17(25): 2805 – 2806.

J. Dufour, X. Dufour, F. Dioury, J. D. Vinko, M easurement of the enthalpy of formation of an iron pico-hydride and of its main properties, Int. J. Mod. Phys. B., 2017, 31(25), 1745007.

2015-2016

Jorge, E.G. ; Rayar, A.M. ; Barigye, S.J. ; Rodriguez, M.E.J. ; Sylla-Iyarreta Veita, M. Development of an in Silico model of DPPH• free radical scavenging capacity: prediction of antioxidant activity of coumarin type compounds. Int. J. Mol. Sci., 2016, 17, 881 (Open access).

Sylla-Iyarreta Veitia M. and Ferroud C. New activation methods used in green chemistry for the synthesis of high value added molecules. Int. J. Energy Environ. Eng. 2015, 6, 37-46.

Renouard S., Corbin C., Colas C., Fidel T., Lopez T., Leclerc E.A., Hendrawati O., Falguières A., Doussot J., Ferroud C., Maunit B., Lainé E. and Hano C. Aerial part of Callitris species as a rich source of deoxypodophyllotoxin. Ind. Crops Prod., 2015, 63, 53-57.

Rayar A., Sylla-Iyarreta Veitia M., Ferroud C. An efficient and selective microwave-assisted Claisen-Schmidt reaction for the synthesis of functionalizedbenzalacetones. Springerplus, 2015, 4, 221 (Open access).

Görmen M., Sylla-Iyarreta Veitia M., Trigui F., El Arbi M., Ferroud C. Ferrocenyl derivatives of bisacodyl: synthesis and antimicrobial activity. J. Organomet. Chem. 2015, 794, 274-281.