Production scientifique de l'équipe Chimie moléculaire


E. Goya Jorge, C. Rampal, N. Loones, S. J. Barigye, R. Gozalbes, C. Ferroud, M. Sylla-Iyarreta Veitía, R. M. Giner. Targeting the aryl hydrocarbon receptor with a novel set of triarylmethanes European Journal of Medicinal Chemistry, 2020, 207, 112777. DOI : 10.1016/j.ejmech.2020.112777

D. Franchi, Z. Amara, Applications of Sensitized-Semiconductors as Heterogeneous Visible-Light Photocatalysts in Organic SynthesisACS Sustain. Chem. Eng. 2020, just accepted, 10.1021/acssuschemeng.0c05179, Open Access

G. Schwertz, A. Zanetti, M. Nascimento de Oliveira, M. A. Gomez Fernandez, Z. Amara, J. Cossy, Chemo- and Diastereoselective Hydrosilylation of Amorphadiene toward the Synthesis of ArtemisininJ. Org. Chem. 2020, 85, 9607, Open Access

E. Goya-Jorge, F. Abdmouleh, L. E. Carpio, R. M. Giner, M. Sylla-Iyarreta Veitía, Discovery of 2-aryl and 2-pyridinylbenzothiazoles endowed with antimicrobial and aryl hydrocarbon receptor agonistic activities, Eur. J. Pharm. Sci., 2020, 151, 105386, DOI : 10.1016/j.ejps.2020.105386

E. Goya-Jorge, R. M. Giner, M. Sylla-Iyarreta Veitía, R. Gozalbes, S. J. Barigye, Predictive modeling of aryl hydrocarbon receptor (AhR) agonism, Chemosphere, 2020, 256, 127068. DOI: 10.1016/j.chemosphere.2020.127068

J. C. S. Terra, A. Desgranges, C. Monnereau, E. H. Sanchez, J. A. De Toro, Z. Amara, A. Moores, Photocatalysis Meets Magnetism: Designing Magnetically Recoverable Supports for Visible-Light PhotocatalysisACS Appl. Mater. Interfaces, 202010.1021/acsami.0c06126

M. Russo, Z. Amara, J. Fenneteau, P. Chaumont-Olive, I. Maimouni, P. Tabeling, J. Cossy, Stable Liquid Foams from a New Polyfluorinated SurfactantChem. Commun., 202010.1039/D0CC02182B

D. Fanfone, D. Stanicki, D. Nonclercq, M. Port, L. Vander Elst, S. Laurent, R. N. Muller, S. Saussez, C. Burtea, Molecular Imaging of Galectin-1 Expression as a Biomarker of Papillary Thyroid Cancer by Using Peptide-Functionalized Imaging ProbesBiology20209, 53, Open Access, Special Issue: Molecular Targets and Targeting in Biomedical Sciences 

C. Ricco, F. Abdmoulehab, C. Riccobono, L. Guenineche, F. Martin, E. Goya-Jorge, N. Lagarde, B. Liagre, M. BenAli, C. Ferroud, M. ElArbi, M. Sylla-Iyarreta Veitía, Pegylated Triarylmethanes: Synthesis, Antimicrobial Activity, Anti-proliferative Behavior and in Silico StudiesBioorg. Chem.​​​​ 202096, 103591

A. Zanetti, P. Chaumont-Olive, G. Schwertz, M. Nascimento de Oliveira, M. A. Gomez Fernandez, Z. Amara, J. Cossy, Crystallization-Induced Diastereoisomer Transformation of Dihydroartemisinic Aldehyde with the Betti BaseOrg. Process Res. Dev., 2020, 10.1021/acs.oprd.9b00481, Open Access, Special Issue: "A Taste of Current French Organic Chemistry".

V. Blanchard, Z. Asbai, K. Cottet, G. Boissonnat, M. Port, Z. Amara, Continuous Flow Photo-oxidations Using Supported Photocatalysts on SilicaOrg. Process Res. Dev., 2020, 10.1021/acs.oprd.9b00420, Special Issue: "A Taste of Current French Organic Chemistry".


M. Sylla-Iyarreta Veitía, C. Rampal, C. Ferroud. An Efficient Access to Unsymmetrical Triarylmethanes by Regioselective Friedel-Crafts Hydroxyalkylation. Trends in Organic chemistry, 2019, 20, 1-13

M. Devreux, C. Henoumont, F. Dioury, D. Stanicki, S. Boutry, L. Larbanoix, C. Ferroud, R. N. Muller, S. Laurent, Bimodal Probe for Magnetic Resonance Imaging and Photoacoustic Imaging Based on a PCTA‐Derived Gadolinium(III) Complex and ZW800–1, Eur. J. Inorg. Chem. 2019, 3354–3365

J. Yong-Sang, F. Dioury, V. Meneyrol, I. Ait-Arsa, J-P. Idoumbin, F. Guibbal, J. Patché, F. Gimié, I. Khantalin, J. Couprie, P. Giraud, S. Benard, C. Ferroud, E. Jestin, O. Meilhac, Development, Synthesis, and 68Ga-Labeling of a Lipophilic Complexing Agent for Atherosclerosis PET Imaging, Eur. J. Med. Chem., 2019, 176, 129-134

C. Robic, M. Port, O. Rousseaux, S. Louguet, N. Fretellier, S. Catoen, C. Factor, S. Le Greneur, C. Medina, P. Bourrinet, I. Raynal, J-M. Idée, C. Corot, Physicochemical and Pharmacokinetic Profiles of Gadopiclenol A New Macrocyclic Gadolinium Chelate With High T1 RelaxivityInvest. Radiol., 2019, 54, 475-484

C. Gomez, G. Hallot, A. Pastor, S. Laurent, E. Brun, C. Sicard-Roselli, M. Port, Metallic Bismuth Nanoparticles: Towards a Robust, Productive and Ultrasound Assisted Synthesis from Batch to Flow-Continuous ChemistryUltrason. Sonochem.2019, 56, 167-173

G. Schwertz, A. Zanetti, M. Nascimento de Oliveira, M. A. Gomez Fernandez, F. Dioury, J. Cossy, Z. Amara, Synthesis of Amorpha-4,11-Diene from Dihydroartemisinic AcidTetrahedron2019, 75, 743-748


J. Vitku, L. Kolatorova, C. Ricco , C. Ferroud , O. Hennebert, T. Skodova , J. Heracek, L. Starka, The Quantitation of 7β-Hydroxy-Epiandrosterone in the Plasma and Seminal Plasma of Men With Different Degrees of Fertility, Physiol. Res. 201867 (Suppl. 3): S511-S519,

L. Halby, N. Marechal, D. Pechalrieu, V. Cura, D-M. Franchini, C. Faux, F. Alby, N. Troffer-Charlier, S. Kudithipudi, A. Jeltsch, W. Aouadi, E. Decroly, J-C. Guillemot, P. Page, C. Ferroud, L. Bonnefond, D. Guianvarc’h, J. Cavarelli, P. B. Arimondo, Hijacking DNA methyltransferase transition state analogues to produce chemical scaffolds for PRMT inhibitors. Phil. Trans. R. Soc. B, 2018, 373: 20170072

C. Gomez, G. Hallot, M. Port, Chapter 10, Bismuth metallic nanoparticles, in Inorganic Frameworks as Smart Nanomedicines, edited by Alexandru Mihai Grumezescu,, William Andrew Publishing, 2018, Pages 449-487, ISBN 9780128136614

B. Tambosco, K. Segura, C. Seyrig, D. Cabrera, M. Port, C. Ferroud, Z. Amara, Outer-sphere effects in visible-light photochemical oxidations with immobilized and recyclable ruthenium bipyridyl salts. ACS Catalysis20188, 4383-4389

S. Drouet, B. Haider Abbas, A. Falguières, W. Ahmad, S. Khan, C. Ferroud, J. Doussot, J. R. Vanier, E. Lainé, C. Hano, Single Laboratory Validation of a Quantitative Core Shell-Based LC Separation for the Evaluation of Silymarin Variability and Associated Antioxidant Activity of Pakistani Ecotypes of Milk Thistle (Silybum Marianum L.). Molecules, 2018, 23, 904

A. Rayar, N. Lagarde, F. Martin, F. Blanchard, B. Liagre, C. Ferroud, J-F Zagury, M. Montes, M. Sylla-Iyarreta Veitía, New selective cyclooxygenase-2 inhibitors from cyclocoumarol: synthesis, characterization, biological evaluation and molecular modeling. Eur. J. Med. Chem., 2018, 146, 577-587


D. Siverio-Mota, I. Andujar, Y. Marrero-Ponce, R. M. Giner, C. Díaz Mendoza, G. Manjarrez Paba, L. Vicet-Muro, M. L. Cordero-Maldonado, P. A. M de Witte, A. D. Crawford, M. Sylla-Iyarreta Veitía, F. Pérez-Jiménez, V. J. Aran. Anti-Inflammatory activity and cheminformatics analysis of new potent 2-substituted 1-methyl-5-nitroindazolinones. Curr. Top. Med. Chem., 2017, 17, 3236 - 3248

L. Halby, Y. Menon, E. Rilova, D. Pechalrieu, V. Masson, C. Faux, M.A. Bouhlel, M-H. David-Cordonnier, N. Novosad, Y. Aussagues, A. Samson, L. Lacroix, F. Ausseil, L. Fleury, D. Guianvarc'h, C. Ferroud, P. Arimondo, Rational design of bisubstrate-type analogs as inhibitors of DNA methyltransferases in cancer cells,  J. Med. Chem.2017, 60, 4665-4679

J. Jin, S. Guidi, Z. Abada, Z. Amara, M. Selva, M. W. George, M. Poliakoff, Continuous niobium phosphate catalysed Skraup reaction for quinoline synthesis from solketal, Green Chem. 2017, 19, 2439-2447

D. S. Lee, Z. Amara, C. A. Clark, Z. Xu, B. Kakimpa, H. P. Morvan, S. J. Pickering, M. Poliakoff, M. W. George, Continuous photo-oxidation in a vortex reactor: efficient operations using air drawn from the laboratory, Org. Process Res. Dev. 2017, 21, 1042-1050

M. Sylla-Iyarreta Veitía, D. Siverio Mota, V. Lerari, M. Marín, R. M. Giner, L. Vicet Muro, Y. Rivero Guerra, F. Dumas, C. Ferroud, P. A. M. de Witte, A. D. Crawford, V. J. Arán, Y. Marrero Ponce, Fishing Anti-Inflammatories from Known Drugs: In Silico Repurposing, Design, Synthesis and Biological Evaluation of Bisacodyl Analogues, Curr. Top. Med. Chem., 2017, 17, 2866 – 2887,

Rayar A.-M., Lagarde N., Ferroud C., Zagury J.-F., Montes M., Sylla-Iyarreta Veitía M., Update on COX-2 Selective Inhibitors: Chemical Classification, Side Effects and their Use in Cancers and Neuronal Diseases, Curr. Top. Med. Chem., 2017, 17, 1-22.

M. Sylla-Iyarreta Veitía, F. Dumas, A. Duardo-Sánchez, S. Arrasate, Editorial: New Experimental and Computational Tools for Drug Discovery: From Chemistry to Biology. Part-III, Curr. Top. Med. Chem, 2017, 17(30): 3234 – 3235.

M. Sylla-Iyarreta Veitía, F. Dumas, H. González-Díaz. Editorial: New Experimental and Computational Tools for Drug Discovery: From Chemistry to Biology. Part-II, Curr. Top. Med. Chem., 2017, 17(26): 2901 – 2902.

M. Sylla-Iyarreta Veitía, F. Dumas, H. González-Díaz, Editorial: New Experimental and Computational Tools for Drug Discovery: From Chemistry to Biology. Part-I, Curr. Top. Med. Chem., 2017, 17(25): 2805 – 2806.


Jorge, E.G. ; Rayar, A.M. ; Barigye, S.J. ; Rodriguez, M.E.J. ; Sylla-Iyarreta Veita, M. Development of an in Silico model of DPPH• free radical scavenging capacity: prediction of antioxidant activity of coumarin type compounds. Int. J. Mol. Sci., 2016, 17, 881 (Open access).

Sylla-Iyarreta Veitia M. and Ferroud C. New activation methods used in green chemistry for the synthesis of high value added molecules. Int. J. Energy Environ. Eng. 2015, 6, 37-46.

Renouard S., Corbin C., Colas C., Fidel T., Lopez T., Leclerc E.A., Hendrawati O., Falguières A., Doussot J., Ferroud C., Maunit B., Lainé E. and Hano C. Aerial part of Callitris species as a rich source of deoxypodophyllotoxin. Ind. Crops Prod., 2015, 63, 53-57.

Rayar A., Sylla-Iyarreta Veitia M., Ferroud C. An efficient and selective microwave-assisted Claisen-Schmidt reaction for the synthesis of functionalizedbenzalacetones. Springerplus, 2015, 4, 221 (Open access).

Görmen M., Sylla-Iyarreta Veitia M., Trigui F., El Arbi M., Ferroud C. Ferrocenyl derivatives of bisacodyl: synthesis and antimicrobial activity. J. Organomet. Chem. 2015, 794, 274-281.